Slow Binding Inhibitors
Robert A. Copeland · 2013
This chapter contains sections titled: Key Learning Points Determining kobs: The Rate Constant for Onset of Inhibition Mechanisms of Slow Binding Inhibition Determination of Mechanism and Assessment of True Affinity Determining Inhibition Modality for Slow Binding Inhibitors SAR for Slow Binding Inhibitors Some Examples of Pharmacologically Interesting Slow Binding Inhibitors Summary References